SCHEMBL13136392

SCHEMBL13136392

Cc1ccnc(Nc2cccc(-c3cnc(N4CCNCC4)s3)n2)c1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KARS1 Q15046 13/20 0.64
SYK P43405 1/20 0.47
CHEK1 O14757 4/20 0.46
DPP4 P27487 1/20 0.46
MAP3K12 Q12852 1/20 0.45
CDK7 P50613 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860076 0.89 KARS1 (0.50) KARS1SYK
SCHEMBL13136401 0.89 KARS1 (0.50) KARS1SYK
SCHEMBL2860446 0.88 KARS1 (0.49) KARS1SYKCHEK1
SCHEMBL13136530 0.88 KARS1 (0.52) KARS1SYK
SCHEMBL2861431 0.86 KARS1 (0.55) KARS1SYK
SCHEMBL13136527 0.86 KARS1 (0.51) KARS1SYKMAP3K12
SCHEMBL13136395 0.85 KARS1 (0.49) KARS1SYK
SCHEMBL2868255 0.85 KARS1 (0.48) KARS1SYKCHEK1
SCHEMBL13136398 0.85 KARS1 (0.48) KARS1SYKCHEK1
SCHEMBL2864564 0.85 SYK (0.51) KARS1SYKCHEK1MAP3K12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7803801-B2 Aminopyridine compounds having Syk inhibitory activity JAPAN TOBACCO, INC. (JP) 2010-09-28 US disclosed
US-7803801-B2 Aminopyridine compounds having Syk inhibitory activity JAPAN TOBACCO, INC. (JP) 2010-09-28 US disclosed
EP-1854793-A1 NOVEL AMINOPYRIDINE COMPOUND WITH Syk INHIBITORY ACTIVITY Japan Tobacco, Inc. (JP) 2007-11-14 EP disclosed