SCHEMBL13152304

SCHEMBL13152304

CCn1c(-c2ccc(N)cc2)c(N)c2ccc(OC(C)C)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK2 Q13002 3/20 0.40
GRIK1 P39086 1/20 0.40
RORC P51449 4/20 0.38
KDM4E B2RXH2 4/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPK1 P28482 2/20 0.36
HTT P42858 2/20 0.36
HSD17B10 Q99714 2/20 0.36
BRD4 O60885 1/20 0.36
BRPF1 P55201 1/20 0.36
HPGD P15428 3/20 0.36
MAPT P10636 3/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CASR P41180 1/20 0.34
MEN1 O00255 1/20 0.33
HBB P68871 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
S1PR3 Q99500 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12109159 0.89 GRIK2 (0.39) GRIK2GRIK1KDM4EALDH1A1MAPK1
SCHEMBL10252659 0.86 GRIK2 (0.54) GRIK2GRIK1KDM4EALDH1A1MAPK1
SCHEMBL10095918 0.85 GRIK2 (0.39) GRIK2GRIK1RORCKDM4EALDH1A1
SCHEMBL13152314 0.84 ALDH1A1 (0.41) RORCKDM4EALDH1A1HPGDMAPT
SCHEMBL13152272 0.81 GRIK2 (0.39) GRIK2GRIK1KDM4EALDH1A1MAPK1
SCHEMBL10249495 0.81 KMT2A (0.46) RORCKDM4EALDH1A1MAPK1HTT
SCHEMBL13152405 0.81 HPGD (0.42) RORCKDM4EALDH1A1MAPK1HTT
SCHEMBL10254357 0.81 ALDH1A1 (0.40) KDM4EALDH1A1MAPK1HTTHSD17B10
SCHEMBL13152111 0.81 GRIK2 (0.38) GRIK2GRIK1KDM4EALDH1A1MAPK1
SCHEMBL13151837 0.81 GRIK2 (0.41) GRIK2GRIK1KDM4EALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118009-A1 HCV INHIBITOR AND THERAPEUTIC AGENT COMBINATIONS PTC THERAPEUTICS, INC. (US) 2010-10-14 WO disclosed