SCHEMBL131548

SCHEMBL131548

COc1cc(CO)cc2c1C(Cc1ccc(-c3ccccc3CO)cc1)NCC2

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.48
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
ADRB3 P13945 1/20 0.48
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL130524 0.93 BCHE (0.51) BCHEADRB2ADRB1ADRB3KDM4E
SCHEMBL131671 0.87 BCHE (0.45) BCHEADRB2ADRB1ADRB3KDM4E
Hydrochloric Acid SCHEMBL145663 0.81 BCHE (0.46) BCHEADRB2ADRB1ADRB3KDM4E
SCHEMBL14172521 0.73 BCHE (0.54) BCHEADRB2ADRB1ADRB3KDM4E
SCHEMBL190641 0.71 BCHE (0.43) BCHEADRB2ADRB1ADRB3KDM4E
SCHEMBL3546894 0.71 BCHE (0.74) BCHEADRB2ADRB1ADRB3KDM4E
SCHEMBL13344580 0.71 BCHE (0.74) BCHEADRB2ADRB1ADRB3KDM4E
SCHEMBL6380551 0.71 BCHE (0.54) BCHEKDM4EMAPTPKM
SCHEMBL14307357 0.71 BCHE (0.74) BCHEADRB2ADRB1ADRB3KDM4E
Hydrochloric Acid SCHEMBL149399 0.71 BCHE (0.42) BCHEADRB2ADRB1ADRB3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120059032-A1 1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES EFFECTIVE AS ANTIGLIOMA AGENTS, METHODS OF MAKING, AND THEIR USE UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2012-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059032-A1 1,2,3,4-TETRAHYDROISOQUINOLINE DERIVATIVES EFFECTIVE AS ANTIGLIOMA AGENTS, METHODS OF MAKING, AND THEIR USE BAD, BAK1, CASP3 BCHE 1788/4885ADRB2 3416/4885ADRB1 3764/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.