SCHEMBL13166111

SCHEMBL13166111

CC(O)c1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4ccccn4)CCOC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTRA1 Q92743 2/20 0.37
DDR2 Q16832 2/20 0.35
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
BDKRB1 P46663 1/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
GRM4 Q14833 1/20 0.33
GSK3B P49841 1/20 0.33
HDAC1 Q13547 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CXCR2 P25025 1/20 0.33
KDR P35968 1/20 0.33
SCN9A Q15858 1/20 0.32
POLB P06746 1/20 0.32
ACACB O00763 1/20 0.32
ROS1 P08922 1/20 0.32
ALK Q9UM73 1/20 0.32
P2RX7 Q99572 1/20 0.32
MMP1 P03956 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13165721 0.96 HTRA1 (0.36) HTRA1DDR2HPGDMAPK1BDKRB1
SCHEMBL765827 0.92 BDKRB1 (0.39) HTRA1DDR2HPGDMAPK1BDKRB1
SCHEMBL13165804 0.90 P2RX7 (0.40) HTRA1DDR2BDKRB1GRM4ALDH1A1
SCHEMBL13166110 0.89 MAPK14 (0.39) HPGDBDKRB1CXCR2SCN9A
SCHEMBL13165771 0.88 DDR2 (0.35) DDR2BDKRB1SCN9A
SCHEMBL13165723 0.88 BDKRB1 (0.35) DDR2MAPK1BDKRB1SCN9AACACB
SCHEMBL13165722 0.87 SCN9A (0.35) DDR2SCN9APOLBMMP1MMP13
SCHEMBL13165774 0.87 DDR2 (0.38) DDR2BDKRB1GRM4SCN9APOLB
SCHEMBL13165595 0.87 BDKRB1 (0.39) HPGDMAPK1BDKRB1SCN9APOLB
SCHEMBL13165726 0.86 BDKRB1 (0.41) DDR2BDKRB1SCN9AACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed