SCHEMBL13166114

SCHEMBL13166114

CC(O)c1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4cn(C)cn4)CCOCC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.43
DDR2 Q16832 2/20 0.35
BDKRB1 P46663 2/20 0.33
SLC6A9 P48067 3/20 0.33
KCNH2 Q12809 3/20 0.33
CYP3A4 P08684 2/20 0.33
SLC6A5 Q9Y345 1/20 0.33
CXCR2 P25025 1/20 0.32
SCN9A Q15858 1/20 0.31
ALK Q9UM73 3/20 0.31
RAF1 P04049 2/20 0.31
ROS1 P08922 1/20 0.31
TP53 P04637 1/20 0.31
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
MAPT P10636 1/20 0.31
CYP2D6 P10635 1/20 0.31
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764459 0.96 GRM2 (0.45) GRM2DDR2BDKRB1SLC6A9KCNH2
SCHEMBL13165808 0.90 GRM2 (0.41) GRM2DDR2BDKRB1TP53MAPT
SCHEMBL13165721 0.88 HTRA1 (0.36) DDR2BDKRB1CXCR2SCN9AALK
SCHEMBL13166115 0.87 DDR2 (0.36) GRM2DDR2BDKRB1CXCR2SCN9A
SCHEMBL13165719 0.86 SCN9A (0.36) BDKRB1SCN9AUBE2MDCUN1D1MAPT
SCHEMBL13166050 0.85 GRM2 (0.40) GRM2DDR2BDKRB1SLC6A9KCNH2
SCHEMBL13165672 0.85 BDKRB1 (0.36) DDR2BDKRB1SCN9AMAPTOPRL1
SCHEMBL13165713 0.85 MAPK14 (0.40) BDKRB1CXCR2SCN9AUBE2MDCUN1D1
SCHEMBL12238934 0.85 GRM2 (0.43) GRM2DDR2BDKRB1SLC6A9KCNH2
SCHEMBL13165730 0.85 BDKRB1 (0.43) BDKRB1KCNH2CXCR2SCN9ARAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed