SCHEMBL764459

SCHEMBL764459

CC(O)c1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4cn(C)cn4)CC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.45
DDR2 Q16832 2/20 0.36
BDKRB1 P46663 3/20 0.35
SLC6A9 P48067 5/20 0.34
KCNH2 Q12809 4/20 0.34
CYP3A4 P08684 2/20 0.34
SLC6A5 Q9Y345 2/20 0.34
PSMB11 A5LHX3 1/20 0.33
PSMA7 O14818 1/20 0.33
PSMB1 P20618 1/20 0.33
PSMA1 P25786 1/20 0.33
PSMA2 P25787 1/20 0.33
PSMA3 P25788 1/20 0.33
PSMA4 P25789 1/20 0.33
PSMB8 P28062 1/20 0.33
PSMB9 P28065 1/20 0.33
PSMA5 P28066 1/20 0.33
PSMB4 P28070 1/20 0.33
PSMB6 P28072 1/20 0.33
PSMB5 P28074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13166114 0.96 GRM2 (0.43) GRM2DDR2BDKRB1SLC6A9KCNH2
SCHEMBL12238934 0.89 GRM2 (0.43) GRM2DDR2BDKRB1SLC6A9KCNH2
SCHEMBL765827 0.86 BDKRB1 (0.39) DDR2BDKRB1PSMB11PSMA7PSMB1
SCHEMBL765174 0.85 DDR2 (0.38) GRM2DDR2BDKRB1PSMB11PSMA7
SCHEMBL764434 0.85 DDR2 (0.38) DDR2BDKRB1PSMB11PSMA7PSMB1
SCHEMBL10121197 0.85 DDR2 (0.41) DDR2BDKRB1HTR2A
SCHEMBL13165808 0.85 GRM2 (0.41) GRM2DDR2BDKRB1TP53
SCHEMBL765640 0.84 SCN9A (0.38) DDR2BDKRB1CYP3A4PSMB11PSMA7
SCHEMBL764500 0.83 BDKRB1 (0.43) BDKRB1PSMB11PSMA7PSMB1PSMA1
SCHEMBL13165721 0.83 HTRA1 (0.36) DDR2BDKRB1SCN9AALKROS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188254-B1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2012-03-21 EP disclosed