SCHEMBL13166115

SCHEMBL13166115

CC(O)c1ccc(Oc2ccc(CNC(=O)C3(NC(=O)c4nccn4C)CCOCC3)cc2)c(C(F)(F)F)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DDR2 Q16832 2/20 0.36
BDKRB1 P46663 2/20 0.33
AR P10275 2/20 0.33
ALK Q9UM73 3/20 0.32
ROS1 P08922 1/20 0.32
EPHX2 P34913 1/20 0.32
CXCR2 P25025 1/20 0.32
CHRNA7 P36544 1/20 0.31
SCN9A Q15858 1/20 0.31
RAF1 P04049 2/20 0.31
GRM2 Q14416 1/20 0.31
TP53 P04637 1/20 0.31
GRM4 Q14833 1/20 0.31
CYP2D6 P10635 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13165774 0.96 DDR2 (0.38) DDR2BDKRB1ARALKROS1
SCHEMBL764434 0.95 DDR2 (0.38) DDR2BDKRB1ARALKROS1
SCHEMBL13165811 0.90 P2RX7 (0.38) DDR2BDKRB1EPHX2KDM4EPOLB
SCHEMBL13166114 0.87 GRM2 (0.43) DDR2BDKRB1ALKROS1CXCR2
SCHEMBL13165672 0.87 BDKRB1 (0.36) DDR2BDKRB1SCN9AMAPT
SCHEMBL13165721 0.86 HTRA1 (0.36) DDR2BDKRB1ALKROS1CXCR2
SCHEMBL13165719 0.86 SCN9A (0.36) BDKRB1SCN9APOLBMAPT
SCHEMBL13166049 0.85 DDR2 (0.38) DDR2EPHX2KDM4EPOLBMAPT
SCHEMBL13165713 0.85 MAPK14 (0.40) BDKRB1EPHX2CXCR2SCN9A
SCHEMBL13165730 0.85 BDKRB1 (0.43) BDKRB1CXCR2SCN9ARAF1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097374-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed