SCHEMBL13183458

SCHEMBL13183458

Cc1ccccc1C1=NNC(=O)C1(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3A Q14432 18/20 0.45
PDE4B Q07343 16/20 0.45
PDE3B Q13370 2/20 0.45
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
THRB P10828 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
CASP1 P29466 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
CASP7 P55210 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380645 0.77 PDE3A (0.54) PDE3APDE4BPDE3BMEN1ALDH1A1
SCHEMBL2840727 0.73 PDE3A (0.40) PDE3APDE4BPDE3B
SCHEMBL6563643 0.72 PDE3A (0.42) PDE3APDE4BPDE3B
SCHEMBL11101816 0.69 NPC1 (0.45) KDM4EMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL2844398 0.67 PDE3A (0.45) PDE3APDE4BPDE3B
SCHEMBL16150403 0.67 PDE3A (0.55) PDE3APDE4BPDE3B
SCHEMBL2847376 0.67 PDE3A (0.55) PDE3APDE4BPDE3B
SCHEMBL16150009 0.67 PDE3A (0.55) PDE3APDE4BPDE3BMEN1ALDH1A1
SCHEMBL2847233 0.66 PDE3A (0.57) PDE3APDE4BPDE3B
SCHEMBL5183107 0.66 PDE3A (0.44) PDE3APDE4BPDE3BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010110400-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2010-09-30 WO disclosed