SCHEMBL13190099

SCHEMBL13190099

CC(F)(F)c1cc2c(cc1C(=O)O)[C@H](NC(=O)c1ccccc1Cl)CCO2

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.45
ALDH1A1 P00352 1/20 0.43
TAS1R3 Q7RTX0 3/20 0.39
TAS1R1 Q7RTX1 3/20 0.39
TAS1R2 Q8TE23 3/20 0.39
BDKRB1 P46663 4/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
BRD4 O60885 2/20 0.39
CREBBP Q92793 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM6B O15054 2/20 0.38
KDM4C Q9H3R0 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2819085 0.92 HSD17B2 (0.46) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL2819081 0.92 HSD17B2 (0.46) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL13190089 0.91 HSD17B2 (0.44) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL2816141 0.85 ALDH1A1 (0.47) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL2816139 0.85 ALDH1A1 (0.47) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL2817719 0.84 HSD17B2 (0.47) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL2817718 0.84 HSD17B2 (0.47) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL784603 0.79 ALDH1A1 (0.50) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL784602 0.79 ALDH1A1 (0.50) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL784976 0.79 ALDH1A1 (0.49) ALDH1A1TAS1R3TAS1R1TAS1R2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed