SCHEMBL13190089

SCHEMBL13190089

COC(=O)c1cc2c(cc1C(C)(F)F)OCC[C@H]2NC(=O)c1ccccc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.44
ALDH1A1 P00352 2/20 0.42
SPTLC2 O15270 1/20 0.39
TAS1R3 Q7RTX0 6/20 0.38
TAS1R1 Q7RTX1 6/20 0.38
TAS1R2 Q8TE23 6/20 0.38
MAPT P10636 3/20 0.38
BRD4 O60885 2/20 0.38
CREBBP Q92793 2/20 0.38
BDKRB1 P46663 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
TP53 P04637 1/20 0.36
POLB P06746 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TRPV1 Q8NER1 2/20 0.36
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2817718 0.94 HSD17B2 (0.47) HSD17B2ALDH1A1SPTLC2TAS1R3TAS1R1
SCHEMBL2817719 0.94 HSD17B2 (0.47) HSD17B2ALDH1A1SPTLC2TAS1R3TAS1R1
SCHEMBL13190099 0.91 HSD17B2 (0.45) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL15235419 0.87 ALDH1A1 (0.45) HSD17B2ALDH1A1SPTLC2TAS1R3TAS1R1
SCHEMBL2819081 0.83 HSD17B2 (0.46) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL2819085 0.83 HSD17B2 (0.46) HSD17B2ALDH1A1TAS1R3TAS1R1TAS1R2
SCHEMBL803721 0.81 SPTLC2 (0.49) HSD17B2ALDH1A1SPTLC2TAS1R3TAS1R1
SCHEMBL485049 0.81 ALDH1A1 (0.47) ALDH1A1SPTLC2TAS1R3TAS1R1TAS1R2
SCHEMBL784581 0.81 ALDH1A1 (0.47) ALDH1A1SPTLC2TAS1R3TAS1R1TAS1R2
SCHEMBL2816141 0.77 ALDH1A1 (0.47) HSD17B2ALDH1A1SPTLC2TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed