SCHEMBL13194

SCHEMBL13194

CCOC(=O)c1nn(-c2cccc(NC(=O)N3CCOCC3)c2)c2c1C[S+]([O-])c1ccccc1-2

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 17/20 0.54
PIK3R2 O00459 17/20 0.54
PIK3CA P42336 17/20 0.54
PIK3CB P42338 17/20 0.54
PIK3CG P48736 17/20 0.54
PIK3R5 Q8WYR1 17/20 0.54
PIK3R3 Q92569 17/20 0.54
RAB9A P51151 2/20 0.44
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13037 0.89 PIK3CD (0.59) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL12276251 0.83 PIK3CD (0.79) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL13078 0.81 PIK3CD (0.53) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL13184 0.81 ALDH1A1 (0.51) RAB9AALDH1A1NPC1
SCHEMBL12904 0.81 ALDH1A1 (0.44) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL18082699 0.81 ALDH1A1 (0.46) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL18082720 0.80 PIK3CD (0.52) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL18082703 0.80 PIK3CD (0.43) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG
SCHEMBL18082643 0.80 ALDH1A1 (0.48) ALDH1A1SMN1; SMN2NPC1
SCHEMBL18082839 0.79 PIK3CD (0.49) PIK3CDPIK3R2PIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058149-A1 TRICYCLIC PYRAZOL AMINE DERIVATIVES MERCK SERONO S.A. (CH) 2011-05-19 WO disclosed