SCHEMBL13208366

SCHEMBL13208366

CPNc1ccc2c(Oc3ccc(F)cc3)cccc2n1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NCF1 P14598 4/20 0.43
SCN9A Q15858 10/20 0.41
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2907740 0.76 CYP1A2 (0.52) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL1616630 0.76 SCN9A (0.43) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL1615592 0.71 PFKFB3 (0.42)
SCHEMBL1616049 0.69 LMNA (0.48) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL16717433 0.67 ADORA1 (0.52) KDM4ECYP1A2MAPTLMNAMEN1
SCHEMBL27303568 0.66 KDR (0.49) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL3697880 0.66 MAPT (0.51) KDM4ECYP1A2MAPTCYP2C9CYP2C19
SCHEMBL27060737 0.65 NCF1 (0.65) KDM4ECYP1A2CYP2C19TDP1NCF1
SCHEMBL21217198 0.65 NCF1 (0.53) KDM4EMAPTTDP1NCF1LMNA
Hydrochloric Acid SCHEMBL27300484 0.65 MAPT (0.50) KDM4ECYP1A2MAPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099763-B1 2-AMINOQUINOLINES AS 5-HT(5A) RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-08-11 EP disclosed