SCHEMBL13255449

SCHEMBL13255449

Oc1c(-c2nnc(Cc3ccc(F)cc3)s2)oc2cccnc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.40
POLB P06746 2/20 0.37
PARP1 P09874 1/20 0.37
KDM4E B2RXH2 4/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
RAB9A P51151 3/20 0.36
HPGD P15428 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
HDAC6 Q9UBN7 1/20 0.34
KMT2A Q03164 5/20 0.34
MEN1 O00255 4/20 0.34
NPC1 O15118 2/20 0.33
BCHE P06276 1/20 0.33
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
USP2 O75604 1/20 0.32
MAPT P10636 1/20 0.32
ALOX12 P18054 1/20 0.32
MPI P34949 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13255442 0.84 MAPK14 (0.38) MAPK14POLBPARP1L3MBTL1RAB9A
SCHEMBL13255450 0.78 RAB9A (0.48) MAPK14POLBPARP1KDM4EL3MBTL1
SCHEMBL12020169 0.76 MEN1 (0.41) POLBPARP1KDM4ERAB9ASMN1; SMN2
SCHEMBL13255593 0.70 PARP1 (0.40) MAPK14POLBPARP1KDM4EL3MBTL1
SCHEMBL13255451 0.64 HPGD (0.47) MAPK14POLBKDM4EL3MBTL1RAB9A
SCHEMBL13255381 0.64 MEN1 (0.36) POLBHPGDSMN1; SMN2HDAC6KMT2A
SCHEMBL14046419 0.63 HDAC6 (0.35) POLBRAB9AHPGDHDAC6KMT2A
SCHEMBL13851051 0.62 KMT2A (0.49) L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL13255478 0.61 HPGD (0.47) POLBKDM4EL3MBTL1RAB9AHPGD
SCHEMBL967039 0.61 RAB9A (0.46) POLBKDM4EL3MBTL1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7759372-B2 Nitrogen-containing heteroaryl compounds having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2010-07-20 US disclosed
US-7759372-B2 Nitrogen-containing heteroaryl compounds having inhibitory activity against HIV integrase SHIONOGI & CO., LTD. (JP) 2010-07-20 US disclosed
EP-2033952-A1 Nitrogen-containing Heteroaryl compounds having HIV Integrase Inhibitory Activity Shionogi&Co., Ltd. (JP) 2009-03-11 EP disclosed