SCHEMBL13257972

SCHEMBL13257972

O=C(NCc1ccccc1O)c1ccc2nn(C3CCOCC3)c(=O)n2c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.42
NAMPT P43490 7/20 0.39
ROCK1 Q13464 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.37
MAPK1 P28482 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CHRM4 P08173 1/20 0.36
MAPK8 P45983 1/20 0.36
SPR P35270 1/20 0.36
BRD4 O60885 1/20 0.36
METTL3 Q86U44 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13258579 0.89 ROCK2 (0.40) ROCK2NAMPTROCK1RXFP1KMT2A
SCHEMBL3786977 0.77 EPHX2 (0.47) ROCK2ROCK1
SCHEMBL3795177 0.75 DDR1 (0.43) ROCK2NAMPTROCK1
SCHEMBL3785014 0.74 DDR1 (0.46) NAMPT
SCHEMBL3794531 0.74 ROCK2 (0.47) ROCK2ROCK1BRD4
SCHEMBL13258576 0.72 DDR1 (0.41) ROCK2ROCK1
SCHEMBL13258575 0.72 DDR1 (0.41) ROCK2ROCK1
SCHEMBL3792501 0.66 CNR2 (0.48) ROCK2ROCK1
SCHEMBL5723909 0.64 HPGD (0.67) KMT2AMEN1TSHR
SCHEMBL30646449 0.64 HPGD (0.67) KMT2AMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed