SCHEMBL13258403

SCHEMBL13258403

CCCCOc1nc2[nH]ccc2c(=O)n1-c1ccc(O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
LMNA P02545 4/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
NPY1R P25929 1/20 0.54
NPY2R P49146 1/20 0.54
MAPK1 P28482 3/20 0.44
METAP2 P50579 1/20 0.40
ESR1 P03372 4/20 0.39
ESR2 Q92731 3/20 0.39
LTA4H P09960 2/20 0.37
NR5A1 Q13285 1/20 0.37
MAPT P10636 3/20 0.35
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
RAB9A P51151 2/20 0.35
CYP2C9 P11712 1/20 0.35
TP53 P04637 1/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13257650 0.90 LMNA (0.43) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL2561543 0.85 ALDH1A1 (0.48) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL13257467 0.81 ALDH1A1 (0.34) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL2565275 0.81 PIK3CD (0.46) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL13258448 0.81 JAK1 (0.37)
SCHEMBL13266550 0.79 MAPT (0.43) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL13257678 0.78 PDE11A (0.43) LMNAMAPK1ESR1ESR2MAPT
SCHEMBL2567106 0.78 PIK3CD (0.44) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL2566379 0.76 PIK3CD (0.44) ALDH1A1LMNAL3MBTL1NPY1RNPY2R
SCHEMBL2561251 0.76 PIK3CD (0.47) ALDH1A1LMNAL3MBTL1NPY1RNPY2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010087467-A1 DELTA-5-DESATURASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-05 WO disclosed