SCHEMBL13259451

SCHEMBL13259451

Bc1ccc(N)c(NCCO)c1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.36
PRSS1 P07477 10/20 0.35
CYP2C19 P33261 2/20 0.34
CYP2D6 P10635 1/20 0.34
RECQL P46063 1/20 0.34
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 2/20 0.33
GLA P06280 2/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6657713 0.81 KMT2A (0.37) KMT2APRSS1CYP2C19CYP2D6RECQL
SCHEMBL30461744 0.78 MAPT (0.44) KMT2APRSS1CYP2C19CYP2D6RECQL
SCHEMBL418892 0.78 MAPT (0.44) KMT2APRSS1CYP2C19CYP2D6RECQL
SCHEMBL10099695 0.78 SMN1; SMN2 (0.43) KMT2ACYP2C19CYP2D6TSHRTDP1
SCHEMBL3897070 0.74 ALDH1A1 (0.47) KMT2ARECQLTDP1KDM4EGLA
SCHEMBL20571668 0.74 KDM4E (0.41) KMT2ACYP2C19RECQLKDM4EALDH1A1
SCHEMBL6896833 0.73 KMT2A (0.62) KMT2ATSHRTDP1KDM4EALDH1A1
SCHEMBL30128490 0.72 KDM4E (0.49) KMT2APRSS1CYP2C19CYP2D6RECQL
SCHEMBL7375160 0.72 KDM4E (0.49) KMT2APRSS1CYP2C19CYP2D6RECQL
SCHEMBL13259052 0.71 MAPT (0.54) KMT2ATSHRTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093425-A1 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2010-08-19 WO disclosed