SCHEMBL13273166

SCHEMBL13273166

CCN1C(=O)CCc2cc(-c3ccc(C(F)(F)F)cc3)ccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 5/20 0.60
CYP11B1 P15538 5/20 0.60
CYP1A2 P05177 2/20 0.60
ATAD2 Q6PL18 1/20 0.58
KIF11 P52732 2/20 0.47
HDAC6 Q9UBN7 3/20 0.44
HDAC1 Q13547 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
TDP2 O95551 1/20 0.43
BRD4 O60885 1/20 0.42
BMPR1B O00238 1/20 0.41
BMPR1A P36894 1/20 0.41
TGFBR1 P36897 1/20 0.41
ACVRL1 P37023 1/20 0.41
ACVR1 Q04771 1/20 0.41
NOTUM Q6P988 1/20 0.40
CYP17A1 P05093 1/20 0.40
CYP19A1 P11511 1/20 0.40
MET P08581 1/20 0.39
DGAT1 O75907 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3310122 0.86 BRD4 (0.47) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL3307667 0.84 KIF11 (0.45) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL3309660 0.84 KIF11 (0.45) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL3306413 0.83 KIF11 (0.44) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL13330272 0.83 HSP90AA1 (0.53) CYP11B2CYP11B1CYP1A2HDAC6HDAC1
SCHEMBL3306832 0.82 MET (0.47) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL3310395 0.82 KIF11 (0.43) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL3315684 0.82 HDAC6 (0.44) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL4596531 0.82 GRIN1 (0.46) CYP11B2CYP11B1CYP1A2ATAD2KIF11
SCHEMBL4892413 0.82 CYP11B1 (0.58) CYP11B2CYP11B1CYP1A2KIF11HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO disclosed