SCHEMBL13282525

SCHEMBL13282525

O=C(O)C(CNc1ccccc1)c1cccc(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.48
MTOR P42345 1/20 0.47
KDM4E B2RXH2 1/20 0.47
HDAC4 P56524 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC5 Q9UQL6 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
HPGD P15428 1/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KCNK3 O14649 1/20 0.42
OPRM1 P35372 3/20 0.42
OPRL1 P41146 2/20 0.42
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
SLC6A2 P23975 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13285509 0.84 CYP2C19 (0.50) POLBMAPTMAPK1
SCHEMBL16664416 0.84 MEN1 (0.46) MTORKDM4EPOLBMAPTMAPK1
SCHEMBL30371733 0.80 CNR2 (0.50) CNR2HDAC4HDAC7HDAC5MEN1
SCHEMBL6366263 0.78 HDAC4 (0.49) CNR2HDAC4HDAC7HDAC5MEN1
SCHEMBL6366259 0.78 HDAC4 (0.49) CNR2HDAC4HDAC7HDAC5MEN1
SCHEMBL6366254 0.78 HDAC4 (0.49) CNR2HDAC4HDAC7HDAC5MEN1
SCHEMBL29421137 0.76 AKR1C3 (0.51) CNR2HDAC4HDAC7HDAC5CES2
SCHEMBL27953660 0.76 MEN1 (0.48) CNR2HDAC4HDAC7HDAC5POLB
SCHEMBL2016833 0.76 AKR1C3 (0.51) CNR2HDAC4HDAC7HDAC5CES2
SCHEMBL2864430 0.76 ROCK2 (0.49) CNR2HDAC4HDAC7HDAC5CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072338-A1 ALKALOID AMINOESTER DERIVATIVES AND MEDICINAL COMPOSITION THEREOF CHIESI FARMACEUTICI S.P.A. (IT) 2010-07-01 WO disclosed