SCHEMBL13286252

SCHEMBL13286252

COCc1ccc(C(=O)NCc2ccncc2)cc1-c1ccc(I)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 0.49
GAA P10253 1/20 0.47
ROCK2 O75116 6/20 0.47
ROCK1 Q13464 4/20 0.47
CYP3A4 P08684 4/20 0.47
GSK3B P49841 3/20 0.47
PRKACA P17612 2/20 0.47
GSK3A P49840 2/20 0.47
PRKX P51817 2/20 0.47
CLK4 Q9HAZ1 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
PRKCQ Q04759 1/20 0.47
LMNA P02545 4/20 0.46
RPS6KA5 O75582 1/20 0.46
MAP4K4 O95819 1/20 0.46
PRKCG P05129 1/20 0.46
RPS6KB1 P23443 1/20 0.46
MAPK1 P28482 1/20 0.46
AKT1 P31749 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13285983 0.92 MMP13 (0.49) MMP13GAAROCK2ROCK1CYP3A4
SCHEMBL792267 0.89 CYP3A4 (0.57) MMP13GAAROCK2ROCK1CYP3A4
SCHEMBL13285990 0.81 RAB9A (0.50) ROCK2ROCK1CYP3A4CYP2C9MAPK1
SCHEMBL10283543 0.81 CYP3A4 (0.57) MMP13GAAROCK2ROCK1CYP3A4
SCHEMBL13286253 0.73 CYP3A4 (0.38) ROCK2CYP3A4CLK4CYP2D6MAPK1
SCHEMBL13286177 0.73 HPGD (0.44) MMP13CYP2D6CYP2C9SMN1; SMN2MAPK14
SCHEMBL13285970 0.72 MAPK14 (0.45) GAAROCK2SMN1; SMN2MAPK14ALDH1A1
SCHEMBL30828595 0.72 MMP13 (0.88) MMP13GAAROCK2ROCK1CYP3A4
SCHEMBL13947076 0.71 NR1H4 (0.71) MMP13GAACYP3A4LMNAMAPK1
SCHEMBL13286176 0.71 PLK1 (0.39) ROCK2ROCK1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2206715-A1 Fused heterotetracyclic compounds and use thereof as hcv polymerase inhibitor Japan Tobacco, Inc. (JP) 2010-07-14 EP disclosed