SCHEMBL13286256

SCHEMBL13286256

CCCN(C)C(=O)c1ccc(-c2ccc(I)cc2)c(COC)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 5/20 0.42
TLR9 Q9NR96 2/20 0.36
TLR8 Q9NR97 2/20 0.36
TLR7 Q9NYK1 2/20 0.36
GYS1 P13807 1/20 0.36
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
DRD2 P14416 1/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
HDAC4 P56524 1/20 0.34
HPGD P15428 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
NAMPT P43490 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13286262 0.91 PDK2 (0.40) PDK2TLR9TLR8TLR7GYS1
SCHEMBL792216 0.88 PDK2 (0.42) PDK2GYS1
SCHEMBL13286175 0.84 HSP90AA1 (0.48) PDK2HPGD
SCHEMBL13285989 0.83 KMT2A (0.51) ROCK2ROCK1HPGD
SCHEMBL13286249 0.79 CHEK2 (0.39)
SCHEMBL791690 0.79 PDK2 (0.40) PDK2HDAC4
SCHEMBL792151 0.79 ALDH1A1 (0.44) PDK2HPGD
SCHEMBL13285970 0.78 MAPK14 (0.45) PDK2ROCK2HPGDNAMPT
SCHEMBL13285895 0.77 SMN1; SMN2 (0.31) DRD2
SCHEMBL13286253 0.77 CYP3A4 (0.38) ROCK2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2206715-A1 Fused heterotetracyclic compounds and use thereof as hcv polymerase inhibitor Japan Tobacco, Inc. (JP) 2010-07-14 EP disclosed