SCHEMBL13286262

SCHEMBL13286262

CCN(C)C(=O)c1ccc(-c2ccc(I)cc2)c(COC)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.40
HDAC4 P56524 1/20 0.36
HSP90AA1 P07900 2/20 0.35
HSP90AB1 P08238 2/20 0.35
SRD5A2 P31213 1/20 0.34
HSD17B2 P37059 4/20 0.33
ROCK2 O75116 2/20 0.33
ROCK1 Q13464 2/20 0.33
CYP1A2 P05177 1/20 0.33
BLM P54132 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
TLR9 Q9NR96 1/20 0.33
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
NLRP3 Q96P20 1/20 0.33
GYS1 P13807 2/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13286256 0.91 PDK2 (0.42) PDK2HDAC4ROCK2ROCK1HPGD
SCHEMBL13286175 0.89 HSP90AA1 (0.48) PDK2HSP90AA1HSP90AB1CYP1A2BLM
SCHEMBL791690 0.88 PDK2 (0.40) PDK2HDAC4LMNATSHR
SCHEMBL13285989 0.85 KMT2A (0.51) HSD17B2ROCK2ROCK1HPGDTSHR
SCHEMBL13286249 0.81 CHEK2 (0.39)
SCHEMBL792151 0.80 ALDH1A1 (0.44) PDK2CYP1A2HPGDTSHR
SCHEMBL792216 0.79 PDK2 (0.42) PDK2TSHRGYS1
SCHEMBL13286253 0.79 CYP3A4 (0.38) ROCK2CYP1A2HPGDTSHR
SCHEMBL13286176 0.79 PLK1 (0.39) HSD17B2ROCK2ROCK1HPGDTSHR
SCHEMBL13285969 0.78 ROCK2 (0.36) ROCK2ROCK1CYP1A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2206715-A1 Fused heterotetracyclic compounds and use thereof as hcv polymerase inhibitor Japan Tobacco, Inc. (JP) 2010-07-14 EP disclosed