SCHEMBL13286376

SCHEMBL13286376

O=C(I)NNc1nc(Cl)ncc1[N+](=O)[O-]

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 15/20 0.53
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
MCL1 Q07820 1/20 0.37
PTK2B Q14289 1/20 0.37
GSK3B P49841 2/20 0.36
AURKA O14965 1/20 0.36
GSK3A P49840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3703983 0.80 PIN1 (0.61) PIN1GSK3BAURKAGSK3A
SCHEMBL3708830 0.78 PIN1 (0.49) PIN1MAPTMEN1KMT2AGSK3B
SCHEMBL4867295 0.75 PIN1 (0.61) PIN1GSK3B
SCHEMBL7491353 0.74 MAPT (0.64) PIN1MAPTGSK3BAURKAGSK3A
Alcohol SCHEMBL27702458 0.72 PIN1 (0.55) PIN1MAPTMEN1CYP1A2CYP3A4
SCHEMBL3158536 0.72 PIN1 (0.55) PIN1MAPTMEN1CYP1A2CYP3A4
SCHEMBL1804900 0.72 PIN1 (0.57) PIN1MAPT
SCHEMBL28657847 0.72 PIN1 (0.57) PIN1MAPTCYP3A4CYP2C9GSK3B
SCHEMBL1496408 0.72 PIN1 (0.57) PIN1MAPTGSK3B
SCHEMBL3178372 0.71 PIN1 (0.50) PIN1MAPTCYP3A4CYP2C9GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed