SCHEMBL3703983

SCHEMBL3703983

O=C(NNc1nc(Cl)ncc1[N+](=O)[O-])c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 10/20 0.61
GAA P10253 3/20 0.49
GSK3B P49841 2/20 0.45
AURKA O14965 1/20 0.45
GSK3A P49840 1/20 0.45
ALDH1A1 P00352 1/20 0.44
HTT P42858 2/20 0.43
PTGS2 P35354 1/20 0.43
VCAM1 P19320 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3708830 0.88 PIN1 (0.49) PIN1GAAGSK3BAURKAGSK3A
SCHEMBL13286376 0.80 PIN1 (0.53) PIN1GSK3BAURKAGSK3A
SCHEMBL3808780 0.79 PLK1 (0.64) PIN1GSK3BAURKAGSK3AALDH1A1
SCHEMBL6191165 0.78 PIN1 (0.52) PIN1GSK3BAURKAGSK3AALDH1A1
SCHEMBL3976795 0.76 PIN1 (1.00) PIN1GSK3BAURKAGSK3AALDH1A1
SCHEMBL3811561 0.74 PIN1 (0.67) PIN1GAAGSK3BAURKAGSK3A
SCHEMBL3707444 0.74 PRKCQ (0.52) GAAGSK3BAURKAGSK3A
SCHEMBL3971786 0.73 PIN1 (0.65) PIN1HTTKDM4E
SCHEMBL13788890 0.72 PIN1 (0.63) PIN1GSK3BAURKAGSK3A
SCHEMBL7491353 0.72 MAPT (0.64) PIN1GSK3BAURKAGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed