SCHEMBL13290346

SCHEMBL13290346

Cc1cc(C)c2c(c1)C(=O)NC2=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 4/20 0.47
CDK4 P11802 2/20 0.47
CCND1 P24385 2/20 0.47
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
CCNA1 P78396 1/20 0.47
PARP1 P09874 2/20 0.41
ALDH1A1 P00352 1/20 0.40
ALDH2 P05091 1/20 0.40
ALDH3A1 P30838 1/20 0.40
CES1 P23141 1/20 0.40
ROS1 P08922 1/20 0.39
CDK5 Q00535 1/20 0.39
ACVR1 Q04771 1/20 0.39
LRRK2 Q5S007 1/20 0.39
EGFR P00533 1/20 0.39
PPOX P50336 1/20 0.38
KMT2A Q03164 2/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13290345 1.00 GSK3B (0.47) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL10563285 0.79 GSK3B (0.41) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL17316982 0.79 ALDH1A1 (0.42) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL17317078 0.79 GSK3B (0.41) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL383165 0.76 CDK4 (0.54) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL20954055 0.76 PARP1 (0.39) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL15088598 0.76 GSK3B (0.49) GSK3BCDK4CCND1CCNA2CDK2
SCHEMBL6036547 0.72 ELANE (0.45) ALDH1A1KMT2AMEN1HSD17B10
SCHEMBL12111227 0.72 ELANE (0.50) ALDH1A1KMT2AMEN1HSD17B10
SCHEMBL6904482 0.72 ELANE (0.45) ALDH1A1KMT2AMEN1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107188875-A A kind of Preparation Method And Their Intermediate of substituted benzene phthalein compounds 联化科技股份有限公司 2017-09-22 CN disclosed
US-7745641-B2 Nitrogen-containing heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-06-29 US disclosed
US-20090054407-A1 Nitrogen-containing heterocyclic compound KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054407-A1 Nitrogen-containing heterocyclic compound NR4A1, NR5A2, PRMT8 GSK3B 2696/4885CDK4 423/4885CCND1 1559/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.