SCHEMBL13290390

SCHEMBL13290390

COc1ccc2c(c1)c(CC(=O)NCCCCNC(=O)c1ccc(-c3c4ccc(=O)cc-4oc4cc(O)ccc34)c(C(=O)O)c1)c(C)n2C(O)c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.47
ALB P02768 1/20 0.47
ESR1 P03372 1/20 0.45
SLC5A2 P31639 2/20 0.44
PTGS2 P35354 6/20 0.44
PTGS1 P23219 1/20 0.44
AVPR2 P30518 1/20 0.43
OXTR P30559 1/20 0.43
AVPR1A P37288 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13290392 0.90 CA1 (0.55)
SCHEMBL861064 0.90 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL13290324 0.89 CA1 (0.54)
SCHEMBL860836 0.87 PTGS2 (0.58) FOLH1SLC5A2PTGS2PTGS1
SCHEMBL10148093 0.86 ALB (0.49) FOLH1ALBESR1SLC5A2
SCHEMBL861480 0.86 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL16181473 0.83 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL14731425 0.82 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL861487 0.81 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL861474 0.81 CA12 (0.56) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7736624-B2 derivatives of non-steroidal anti-inflammatory drugs that exhibit selective binding to cyclooxygenase-2 (COX-2) and that comprise functional groups allowing them to be used for medical diagnosis and/or as therapeutic agents; tissue-targeted therapy UNIV VANDERBILT (US) 2010-06-15 US disclosed