SCHEMBL16181473

SCHEMBL16181473

COc1ccc2c(c1)c(CC(=O)NCCCCNC(O)c1ccc(C(=O)O)c(-c3c4ccc(=O)cc-4oc4cc(O)ccc34)c1)c(C)n2C(=O)c1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.53
PTGS1 P23219 2/20 0.53
HRH4 Q9H3N8 1/20 0.52
HDAC3 O15379 3/20 0.51
HDAC1 Q13547 3/20 0.51
HDAC8 Q9BY41 3/20 0.51
HDAC6 Q9UBN7 3/20 0.51
HDAC2 Q92769 1/20 0.51
CA12 O43570 2/20 0.49
CA4 P22748 2/20 0.49
CA9 Q16790 2/20 0.49
APP P05067 1/20 0.49
BCHE P06276 1/20 0.49
ACHE P22303 1/20 0.49
TRPV1 Q8NER1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861480 0.91 PTGS2 (0.56) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL861064 0.88 PTGS2 (0.57) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL861487 0.87 PTGS2 (0.51) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL14731425 0.86 PTGS2 (0.54) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL860836 0.86 PTGS2 (0.58) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL861474 0.85 CA12 (0.56) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL860837 0.85 PTGS2 (0.50) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL860830 0.84 CA12 (0.55) PTGS2PTGS1HRH4CA12CA4
SCHEMBL861702 0.83 CA12 (0.53) PTGS2PTGS1HRH4CA12CA4
SCHEMBL13290390 0.83 FOLH1 (0.47) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8865130-B2 Methods and compositions for diagnostic and therapeutic targeting of COX-2 VANDERBILT UNIVERSITY (US) 2014-10-21 US disclosed