SCHEMBL13301210

SCHEMBL13301210

PCc1ccc2ccccc2c1-c1c(CP)ccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.48
ALDH1A1 P00352 2/20 0.48
CYP2A6 P11509 1/20 0.48
TSHR P16473 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
HPRT1 P00492 2/20 0.44
MAPT P10636 1/20 0.42
HIF1A Q16665 1/20 0.41
CYP1B1 Q16678 1/20 0.41
WDR5 P61964 1/20 0.41
DNMT1 P26358 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13207448 0.92 ALDH1A1 (0.41) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL30367845 0.79 HSD17B10 (0.50) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL30066585 0.79 CYP2A6 (0.50) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL6267184 0.79 CYP2A6 (0.50) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL8050013 0.79 HSD17B10 (0.50) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL15263192 0.77 ALDH1A1 (0.48) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL5691676 0.77 ALDH1A1 (0.48) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL14392713 0.77 ALDH1A1 (0.48) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL30066580 0.77 ALDH1A1 (0.48) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL12807315 0.77 HSD17B10 (0.48) HSD17B10ALDH1A1CYP2A6TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9718823-B2 2, 6-Di-nitrogen-containing substituted purine derivative, and preparation method, pharmaceutical composition and use thereof ZHEJIANG MEDICINE CO., LTD. XINCHANG PHARMACEUTICAL FACTORY (CN) 2017-08-01 US disclosed
US-20160207924-A1 2, 6-Di-Nitrogen-Containing Substituted Purine Derivative, And Preparation Method, Pharmaceutical Composition And Use Thereof ZHEJIANG MEDICINE CO., LTD. XINCHANG PHARMACEUTICAL FACTORY (CN) 2016-07-21 US disclosed
US-8580763-B2 2, 6-dinitrogen-containing substituted purine derivatives, the preparation and uses thereof ZHANGGUI WU (CN) 2013-11-12 US disclosed
US-20100144663-A1 2, 6-Dinitrogen-Containing Substituted Purine Derivatives, The Preparation And Uses Thereof ZHE JIANG MEDICINE CO., LTD. XINCHANG PHARMACEUTICAL FACTORY (CN) 2010-06-10 US disclosed
EP-1529768-B1 Process for the preparation of TCD-alcohol DM OXEA DEUTSCHLAND GMBH (DE) 2007-10-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160207924-A1 2, 6-Di-Nitrogen-Containing Substituted Purine Derivative, And Preparation Method, Pharmaceutical Composition And Use Thereof NUDT1, PNP, SLC29A2 HSD17B10 3968/4885ALDH1A1 693/4885CYP2A6 323/4885
US-20100144663-A1 2, 6-Dinitrogen-Containing Substituted Purine Derivatives, The Preparation And Uses Thereof PNP, NUDT1, DPYD HSD17B10 3467/4885ALDH1A1 254/4885CYP2A6 153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.