SCHEMBL13307474

SCHEMBL13307474

CN(C)C(=O)c1cc(C(=O)O)cc(S(C)(=O)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.50
FYN P06241 1/20 0.50
CYP1A2 P05177 1/20 0.44
LMNA P02545 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.37
TPMT P51580 1/20 0.36
ALDH1A1 P00352 2/20 0.36
GSR P00390 2/20 0.36
KDM1A O60341 1/20 0.36
LOX P28300 1/20 0.35
LOXL2 Q9Y4K0 4/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD11B1 P28845 1/20 0.35
AKR1C3 P42330 1/20 0.35
F10 P00742 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3185974 0.87 LCK (0.64) LCKFYNCYP1A2LMNATPMT
SCHEMBL13307475 0.86 CA5A (0.36) LCKFYNLMNAGPBAR1ALDH1A1
SCHEMBL13307455 0.84 TPMT (0.48) LCKFYNLMNATPMTALDH1A1
SCHEMBL10400071 0.84 TPMT (0.48) LCKFYNLMNATPMTALDH1A1
SCHEMBL18503821 0.82 LCK (0.58) LCKFYNCYP1A2LMNATPMT
SCHEMBL3860285 0.81 CA12 (0.43) LCKFYNCYP1A2GPBAR1ALDH1A1
SCHEMBL7857786 0.79 LCK (0.55) LCKFYNCYP1A2LMNATPMT
SCHEMBL9040506 0.79 ALDH1A1 (0.47) LCKFYNCYP1A2LMNATPMT
SCHEMBL17615073 0.78 GSR (0.36) GPBAR1ALDH1A1GSRKDM1ALOX
SCHEMBL8061100 0.78 CA1 (0.37) CYP1A2GPBAR1GSRKDM1ALOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7727997-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2010-06-01 US disclosed
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease ELAN PHARMACEUTICALS, INC. 2007-09-13 US disclosed
US-7176242-B2 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives ELAN PHARMACEUTICALS, INC. (US) 2007-02-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213316-A1 Compounds that are effective inhibitors of beta-secretase; inhibitors of beta-secretase-mediated cleavage of amyloid precursor proteins; effective inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques; treatment of disorders such as Alzheimer's Disease BACE1, BACE2, APP LCK 4627/4885FYN 2169/4885CYP1A2 3371/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.