SCHEMBL13308554

SCHEMBL13308554

Cc1cc(-c2c(C)nn(Cc3cncs3)c2C)ccc1C#N

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
EGLN2 Q96KS0 1/20 0.33
CNR1 P21554 1/20 0.33
KDM4E B2RXH2 2/20 0.32
S1PR1 P21453 1/20 0.32
CACNA1H O95180 6/20 0.32
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
BRD4 O60885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3063738 0.89 AR (0.45) ARCYP11B1CYP11B2EGLN2KDM4E
SCHEMBL3073239 0.84 AR (0.41) ARCYP11B1CYP11B2CNR1BRD4
SCHEMBL13309136 0.83 L3MBTL1 (0.45) ARCYP11B1CYP11B2EGLN2CNR1
SCHEMBL13308504 0.79 GRIN1 (0.36) ARCYP11B1CYP11B2EGLN2CNR1
SCHEMBL13308386 0.78 AKR1B1 (0.37) AREGLN2CNR1S1PR1BRD4
SCHEMBL13308976 0.77 CNR1 (0.34) ARCYP11B1CYP11B2EGLN2CNR1
SCHEMBL13308619 0.76 POLB (0.45) AREGLN2KDM4ENPSR1
SCHEMBL13308563 0.76 EGLN2 (0.39) ARCYP11B1CYP11B2EGLN2KDM4E
SCHEMBL13309138 0.75 AR (0.38) ARCYP11B1CYP11B2EGLN2CNR1
SCHEMBL13309040 0.75 EGLN2 (0.38) ARCYP11B1CYP11B2EGLN2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2194045-A1 SUBSTITUTED PYRAZOLE DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2010-06-09 EP disclosed