SCHEMBL13309151

SCHEMBL13309151

COc1ccc(Cn2nc(C)c(-c3ccc(C#N)c(C)c3)c2C)cc1[N+](=O)O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
F11 P03951 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
ALDH1A1 P00352 2/20 0.36
S1PR1 P21453 2/20 0.36
CACNA1H O95180 5/20 0.36
PKM P14618 1/20 0.36
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3070056 0.83 ALDH1A1 (0.45) KDM4EALDH1A1PKM
SCHEMBL13308971 0.79 CYP1A2 (0.43) MAPTALDH1A1PKMLMNASMN1; SMN2
SCHEMBL13309112 0.78 MBOAT4 (0.39) CACNA1H
SCHEMBL3069287 0.78 KDM4E (0.45) KDM4ETP53MAPTPTGDR2ALDH1A1
SCHEMBL3069345 0.78 AR (0.39) KDM4ETP53MAPTPTGDR2ALDH1A1
SCHEMBL13308529 0.77 AR (0.41) KDM4EMAPTALDH1A1S1PR1PKM
SCHEMBL13308414 0.77 KDM4E (0.40) KDM4EF11TP53MAPTALDH1A1
SCHEMBL13308619 0.77 POLB (0.45) KDM4EPTGDR2LMNAFNTAFNTB
SCHEMBL13308563 0.76 EGLN2 (0.39) KDM4ETP53MAPTALDH1A1LMNA
SCHEMBL13308598 0.76 HSD17B10 (0.45) KDM4ETP53MAPTALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2194045-A1 SUBSTITUTED PYRAZOLE DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2010-06-09 EP disclosed