SCHEMBL13329969

SCHEMBL13329969

CN(C)c1nc(NCCc2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 8/20 0.57
HRH1 P35367 2/20 0.57
PTGDR Q13258 4/20 0.49
TLR8 Q9NR97 1/20 0.47
TP53 P04637 1/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ACP1 P24666 1/20 0.44
GSK3B P49841 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13329974 0.83 ESR1 (0.44) HRH4HRH1TP53
SCHEMBL13309932 0.81 HRH4 (0.60) HRH4HRH1PTGDRTLR8
SCHEMBL9911093 0.80 PTGDR (0.72) PTGDR
SCHEMBL17407827 0.79 HRH4 (0.80) HRH4HRH1TLR8
SCHEMBL3228726 0.79 HRH4 (0.57) HRH4HRH1PTGDRTLR8MEN1
SCHEMBL13329973 0.74 TLR8 (0.57) HRH4HRH1PTGDRTLR8TP53
SCHEMBL11309305 0.71 MEN1 (0.56) HRH4TP53MEN1KMT2A
SCHEMBL5805069 0.71 HRH4 (0.70) HRH4HRH1TLR8
SCHEMBL28043771 0.71 HRH4 (0.62) HRH4HRH1PTGDRTLR8
SCHEMBL14869428 0.70 CA1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7722893-B2 Use of substitute 2,4-bis (alkylamino) pyrimidines or quinzolines as antimicrobials CIBA SPECIALTY CHEMICALS CORPORATION (US) 2010-05-25 US disclosed
US-7722893-B2 Use of substitute 2,4-bis (alkylamino) pyrimidines or quinzolines as antimicrobials CIBA SPECIALTY CHEMICALS CORPORATION (US) 2010-05-25 US disclosed