SCHEMBL13330780

SCHEMBL13330780

Cc1cc(Cl)c2nc(-c3nc(-c4ccc(C=O)cc4Cl)no3)cn2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HSD11B1 P28845 1/20 0.37
THRB P10828 1/20 0.36
RARA P10276 7/20 0.35
RARB P10826 7/20 0.35
RARG P13631 7/20 0.35
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
PLAT P00750 1/20 0.34
CASP3 P42574 1/20 0.32
ALDH1A3 P47895 2/20 0.32
ALDH3A1 P30838 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3343142 0.85 NPC1 (0.48) NPC1RAB9ATDP1HSD11B1RARA
SCHEMBL3341183 0.80 DPP4 (0.41) NPC1RAB9ATP53HPGDTSHR
SCHEMBL13330845 0.80 HSD11B1 (0.34) NPC1RAB9ATDP1HSD11B1RARA
SCHEMBL3339985 0.79 NPC1 (0.39) NPC1RAB9ATDP1HSD11B1RARA
SCHEMBL3343195 0.73 NPC1 (0.47) NPC1RAB9ATDP1RARARARB
SCHEMBL3343797 0.73 NPC1 (0.46) NPC1RAB9AHPGDTDP1RARA
SCHEMBL3343805 0.73 NPC1 (0.46) NPC1RAB9AHPGDTDP1RARA
SCHEMBL2505933 0.72 NPC1 (0.41) NPC1RAB9AHPGDMAPK1NPSR1
SCHEMBL13303772 0.72 NPC1 (0.41) NPC1RAB9AHPGDTDP1L3MBTL1
SCHEMBL3339344 0.72 DPP4 (0.41) NPC1RAB9ATP53HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010065760-A1 IMIDAZO [1,2A] PYRIDINE DERIVATIVES, THEIR USE AS S1P1 AGONISTS AND METHODS FOR THEIR PRODUCTION EXELIXIS, INC. (US) 2010-06-10 WO disclosed