SCHEMBL13330893

SCHEMBL13330893

CNc1cc2c(cc1Cl)N(c1nc[nH]n1)CC(C(=O)N1CCC(C#N)(Cc3ccc(F)cc3)CC1)O2

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
PROKR1 Q8TCW9 2/20 0.32
FPR2 P25090 1/20 0.32
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
HTR1A P08908 1/20 0.30
ADRA1A P35348 1/20 0.30
MGLL Q99685 1/20 0.30
PIK3CA P42336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3356328 0.90 ALDH1A1 (0.34) ALDH1A1PROKR1FPR2
SCHEMBL3352647 0.90 ALDH1A1 (0.34) ALDH1A1PROKR1FPR2MGLLPIK3CA
SCHEMBL13330897 0.89 ALDH1A1 (0.32) ALDH1A1PROKR1FPR2
SCHEMBL3356345 0.88 ALDH1A1 (0.37) ALDH1A1PROKR1FPR2
SCHEMBL3359564 0.80 ALDH1A1 (0.32) ALDH1A1PROKR1FPR2MGLL
SCHEMBL3353165 0.79 ALDH1A1 (0.35) ALDH1A1PROKR1FPR2JAK2JAK1
SCHEMBL3354404 0.79 ALDH1A1 (0.33) ALDH1A1PROKR1FPR2
SCHEMBL3353857 0.77 ALDH1A1 (0.36) ALDH1A1PROKR1FPR2
SCHEMBL13308355 0.76 MC4R (0.36) ALDH1A1JAK2JAK1
SCHEMBL3358681 0.76 LMNA (0.35) ALDH1A1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068881-A1 NOVEL BENZODIOXANE AND BENZOXAZINE DERIVATIVES USEFUL AS CC CHEMOKINE RECEPTOR LIGANDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-06-17 WO disclosed