SCHEMBL13330902

SCHEMBL13330902

NC1(Cc2ccc(F)cc2)CCN(C(=O)C2CNc3cc(Cl)c(-n4ccnc4)cc3O2)CC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.33
NAMPT P43490 2/20 0.31
LSS P48449 1/20 0.31
CA12 O43570 1/20 0.31
CA9 Q16790 1/20 0.31
KMT2A Q03164 1/20 0.30
MCHR1 Q99705 1/20 0.30
AKT2 P31751 1/20 0.30
NOS2 P35228 1/20 0.30
P2RX7 Q99572 1/20 0.30
TARDBP Q13148 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3354757 0.89 ALDH1A1 (0.34) CYP19A1NAMPTLSSKMT2AMCHR1
SCHEMBL13331642 0.88 PSEN1 (0.36) AKT2
SCHEMBL13331447 0.87 AKT2 (0.34) AKT2TARDBP
SCHEMBL13330711 0.87 PREP (0.34) AKT2TARDBP
SCHEMBL13330873 0.81 NTRK1 (0.34) NAMPT
SCHEMBL3355489 0.80 ALDH1A1 (0.35)
SCHEMBL3355879 0.79 ALDH1A1 (0.36)
SCHEMBL13330872 0.78 PREP (0.33) NAMPTAKT2
SCHEMBL3352607 0.77 PSEN1 (0.36)
SCHEMBL13308393 0.77 CHRM1 (0.35) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068881-A1 NOVEL BENZODIOXANE AND BENZOXAZINE DERIVATIVES USEFUL AS CC CHEMOKINE RECEPTOR LIGANDS FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-06-17 WO disclosed