SCHEMBL13352198

SCHEMBL13352198

COC(=O)[C@H](Cc1cc(OC(=O)OC(C)(C)C)c(OC(=O)OC(C)(C)C)cc1I)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.46
MTNR1B P49286 2/20 0.46
KLK5 Q9Y337 1/20 0.43
TACR1 P25103 2/20 0.41
SCN9A Q15858 2/20 0.40
CTSS P25774 8/20 0.39
CTSK P43235 7/20 0.39
GSTP1 P09211 1/20 0.37
GSTM2 P28161 1/20 0.37
EPHX2 P34913 1/20 0.37
ACE P12821 1/20 0.36
CTSL P07711 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
CTSB P07858 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL584547 0.91 SCN9A (0.49) MTNR1AMTNR1BKLK5TACR1SCN9A
SCHEMBL584495 0.90 SCN9A (0.47) MTNR1AMTNR1BSCN9ACTSSCTSK
SCHEMBL17061439 0.89 MTNR1A (0.46) MTNR1AMTNR1BKLK5TACR1SCN9A
SCHEMBL17071630 0.87 KLK5 (0.43) KLK5TACR1SCN9ACTSSCTSK
SCHEMBL12035787 0.86 MTNR1A (0.46) MTNR1AMTNR1BKLK5TACR1SCN9A
SCHEMBL4651817 0.84 KLK5 (0.41) KLK5TACR1SCN9ACTSSCTSK
SCHEMBL12035495 0.83 KLK5 (0.46) MTNR1AMTNR1BKLK5TACR1SCN9A
SCHEMBL15701998 0.83 KLK5 (0.46) MTNR1AMTNR1BKLK5TACR1SCN9A
SCHEMBL17101171 0.80 MTNR1A (0.51) MTNR1AMTNR1BTACR1SCN9ACTSS
SCHEMBL18833348 0.80 MTNR1A (0.51) MTNR1AMTNR1BTACR1SCN9ACTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9024093-B2 Fluorination of organic compounds PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-05-05 US disclosed
WO-2010059943-A2 FLUORINATION OF ORGANIC COMPOUNDS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-05-27 WO disclosed