SCHEMBL13355237

SCHEMBL13355237

CC1CN(C(=O)c2ccc(N(C)C(=O)c3ccccc3)cc2)CCC(C)(C)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G1B P04054 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45
ACHE P22303 1/20 0.43
CCR5 P51681 1/20 0.43
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAOA P21397 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
PGR P06401 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
NR1H2 P55055 1/20 0.39
NR1H3 Q13133 1/20 0.39
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
SMO Q99835 1/20 0.39
NAMPT P43490 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL162185 0.78 CA12 (0.45) PLA2G1BATG4BACHEKMT2AALDH1A1
SCHEMBL12169333 0.72 NOTUM (0.49)
SCHEMBL13385734 0.72 RECQL (0.50) KMT2AKDM4EALDH1A1HPGDNAMPT
SCHEMBL13355240 0.71 KDM4E (0.48) KMT2AKDM4EALDH1A1HPGDNAMPT
SCHEMBL9928309 0.71 HPGD (0.61) ACHECCR5ALDH1A1HPGD
SCHEMBL13354704 0.70 PGR (0.42) KMT2AKDM4EMAOAPGRALDH1A1
SCHEMBL13079622 0.70 GAA (0.47) KMT2AKDM4EALDH1A1HTT
SCHEMBL12115285 0.70 KMT2A (0.44) KMT2AKDM4EALDH1A1HTT
SCHEMBL4818101 0.70 CRBN (0.56) ACHECCR5ALDH1A1HPGD
SCHEMBL4818087 0.70 CRBN (0.56) ACHECCR5ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1787982-B1 11Beta-Hydroxysteroid dehydrogenase type 1 active compounds HIGH POINT PHARMACEUTICALS LLC (US) 2010-05-12 EP disclosed
US-7700583-B2 Such as [4-(1,3,3-Trimethyl-6-aza-bicyclo[3.2.1]octane-6-carbonyl)-phenyl]carbamic acid tert-butyl ester; for treatment of metabolic syndrome HIGH POINT PHARMACEUTICALS, LLC (US) 2010-04-20 US disclosed