SCHEMBL13376702

SCHEMBL13376702

Bc1cccc(C#Cc2cccc(C#Cc3c(N)nc(N(C)C(=O)OC(C)(C)C)c4ncn(C)c34)c2)c1

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.31
GRM5 P41594 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13376585 0.91 IKBKB (0.37) BRD4GRM5
SCHEMBL12342077 0.90 BRD4 (0.31) BRD4
SCHEMBL2767060 0.89 BRD4 (0.32) BRD4
SCHEMBL12341871 0.89 GRM4 (0.32) BRD4GRM5
SCHEMBL2768127 0.88 GABRA1 (0.33) BRD4
SCHEMBL2766929 0.88 BRD4 (0.31) BRD4
SCHEMBL12341875 0.87 BRD4 (0.30) BRD4
SCHEMBL2766243 0.86 PTGES (0.36) BRD4
SCHEMBL2766241 0.84 CHUK (0.34)
SCHEMBL2767712 0.84 IKBKB (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888584-B1 1, 6 -DIHYDRO- 1,3, 5, 6-TETRAAZA-AS-INDACENE BASED TRICYCLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS COMPRISING SAME AS INHIBITORS OF IKK ENZYME ACTIVITY BRISTOL MYERS SQUIBB CO (US) 2010-04-21 EP disclosed