SCHEMBL13424977

SCHEMBL13424977

O=N/C(=C\C(=O)c1ncccn1)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.34
CTNNB1 P35222 1/20 0.33
WNT3A P56704 1/20 0.33
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
BLM P54132 1/20 0.32
AGER Q15109 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
LMNA P02545 2/20 0.31
NPC1 O15118 1/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
NAPRT Q6XQN6 1/20 0.31
P4HTM Q9NXG6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3307343 0.76 P2RX7 (0.39) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL3307346 0.76 P2RX7 (0.39) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL3307340 0.76 P2RX7 (0.39) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL2320853 0.66 P2RX7 (0.44) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL3309984 0.66 P2RX7 (0.37) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL3309986 0.66 P2RX7 (0.37) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL7574223 0.65 TSHR (0.35) KDM4ETSHR
SCHEMBL31141952 0.65 AKT1 (0.44) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL726451 0.64 P2RX7 (0.46) P2RX7CTNNB1WNT3AKDM4EMAPT
SCHEMBL108190 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010047774-A2 INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS MALATE SYNTHASE, METHODS OF MARKING AND USES THEREOF THE TEXAS A & M UNIVERSITY SYSTEM (US) 2010-04-29 WO disclosed