SCHEMBL13433259

SCHEMBL13433259

COC(=O)c1cccc(-c2ccc(OC)c(CNC(=O)OC(C)(C)C)c2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
HPGD P15428 2/20 0.45
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
APEX1 P27695 1/20 0.43
HTT P42858 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SUCNR1 Q9BXA5 5/20 0.41
TRPV1 Q8NER1 1/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
SCN9A Q15858 4/20 0.40
KDM4A O75164 1/20 0.39
GFER P55789 1/20 0.38
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3418641 0.86 ALDH1A1 (0.45) ALDH1A1HPGDKDM4EMEN1LMNA
SCHEMBL3416346 0.83 PPARG (0.53) ALDH1A1HPGDKDM4EHTTSMN1; SMN2
SCHEMBL4718383 0.82 SCN9A (0.47) ALDH1A1HPGDKDM4EMEN1LMNA
SCHEMBL13433262 0.80 HDAC1 (0.48) KDM4ESMN1; SMN2PPARGPPARDPPARA
SCHEMBL3413999 0.79 EGFR (0.41) ALDH1A1HPGDKDM4ELMNAHTT
SCHEMBL3415307 0.79 PPARD (0.63) ALDH1A1HPGDKDM4EMEN1LMNA
SCHEMBL13433269 0.78 CYP11B1 (0.50) PPARGPPARDPPARADYRK1A
SCHEMBL3415566 0.78 PPARD (0.40) ALDH1A1HPGDKDM4ELMNAHTT
SCHEMBL4722006 0.77 MAPK1 (0.57) ALDH1A1HPGDKDM4EMEN1HTT
SCHEMBL3413967 0.77 BDKRB1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed