SCHEMBL13433262

SCHEMBL13433262

COC(=O)c1ccnc(-c2ccc(OC)c(CNC(=O)OC(C)(C)C)c2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.48
ACACB O00763 1/20 0.47
ACACA Q13085 1/20 0.47
KDM1A O60341 2/20 0.46
KDM4E B2RXH2 1/20 0.45
KDM6B O15054 1/20 0.45
KDM5C P41229 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
KDM2A Q9Y2K7 1/20 0.45
KDM3A Q9Y4C1 1/20 0.45
JMJD6 Q6NYC1 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
CFTR P13569 1/20 0.41
AAK1 Q2M2I8 4/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3416346 0.88 PPARG (0.53) HDAC1KDM4EPPARGPPARDPPARA
SCHEMBL3416551 0.85 HDAC1 (0.50) HDAC1KDM1AKDM4EKDM6BKDM5C
SCHEMBL13433269 0.83 CYP11B1 (0.50) HDAC1KDM1APPARGPPARDPPARA
SCHEMBL3413912 0.82 PPARD (0.42) HDAC1PPARGPPARDPPARASMN1; SMN2
SCHEMBL3415050 0.81 PPARD (0.41) HDAC1PPARGPPARDPPARA
SCHEMBL3414304 0.81 PPARD (0.43) HDAC1PPARGPPARDPPARA
SCHEMBL3417162 0.80 BDKRB1 (0.42) PPARGPPARDPPARASMN1; SMN2
SCHEMBL3416623 0.80 KDM4E (0.41) KDM4EPPARGPPARDPPARASMN1; SMN2
SCHEMBL13433259 0.80 ALDH1A1 (0.45) KDM4EPPARGPPARDPPARASMN1; SMN2
SCHEMBL3413999 0.80 EGFR (0.41) HDAC1KDM4EPPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed
US-7687664-B2 Carboxylic acid derivative, a salt thereof or an ester of them, and medicament comprising it EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-03-30 US disclosed