SCHEMBL13440367

SCHEMBL13440367

Cc1ccc([C@@H]2CN(Cc3ccc(C#N)cc3)CCN2c2ccc(C#N)cc2Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
KDM4E B2RXH2 2/20 0.48
HPGD P15428 1/20 0.48
ALOX12 P18054 1/20 0.48
DRD4 P21917 4/20 0.47
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
KDM1A O60341 1/20 0.45
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PARP1 P09874 2/20 0.38
TNK1 Q13470 2/20 0.38
TNK2 Q07912 1/20 0.38
PDE2A O00408 1/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11958314 0.94 DRD4 (0.45) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL11957997 0.92 ALDH1A1 (0.44) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL11958313 0.92 CNR1 (0.42) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL11980190 0.92 CNR1 (0.42) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL11979781 0.87 CNR1 (0.47) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL11979760 0.87 CNR1 (0.47) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL11958315 0.87 CNR1 (0.47) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL13877764 0.86 KDM1A (0.42) ALDH1A1KDM4EHPGDALOX12DRD4
SCHEMBL13134643 0.86 DRD2 (0.43) ALDH1A1DRD4SIGMAR1CCR2
SCHEMBL14787574 0.86 CNR1 (0.40) ALDH1A1KDM4EHPGDALOX12DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700597-B2 Substituted piperazines as CB1 antagonists SCHERING CORPORATION (US) 2010-04-20 US disclosed