SCHEMBL13440511

SCHEMBL13440511

N=C1NC(c2ccccc2)(c2ccccc2)C(=O)N1CC1CCN(C(=O)C2C[C@H]2c2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.47
HRH3 Q9Y5N1 11/20 0.46
BACE1 P56817 1/20 0.44
PREP P48147 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545591 1.00 SIGMAR1 (0.47) SIGMAR1HRH3BACE1PREP
SCHEMBL7546546 0.83 HRH1 (0.41) SIGMAR1HRH3BACE1
SCHEMBL17715653 0.83 POLB (0.48) SIGMAR1
SCHEMBL7526895 0.83 HRH3 (0.46) SIGMAR1HRH3BACE1PREP
SCHEMBL7571468 0.82 FASN (0.40) SIGMAR1
SCHEMBL7547422 0.81 KMT2A (0.45) SIGMAR1HRH3
SCHEMBL7541789 0.80 KMT2A (0.49)
SCHEMBL7546132 0.80 HSD11B1 (0.47) SIGMAR1
SCHEMBL7548883 0.80 KMT2A (0.44) SIGMAR1
SCHEMBL7574120 0.79 PARP1 (0.42) SIGMAR1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7700603-B2 Heterocyclic aspartyl protease inhibitors SCHERING CORPORATION (US) 2010-04-20 US disclosed