SCHEMBL13442183

SCHEMBL13442183

N#CCc1ccc(-c2cc(OC3CCNCC3)c3cnccc3c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 8/20 0.51
CHUK O15111 7/20 0.51
ROCK1 Q13464 5/20 0.51
LCK P06239 2/20 0.51
TNF P01375 1/20 0.46
AKT1 P31749 1/20 0.43
MKNK1 Q9BUB5 2/20 0.41
MKNK2 Q9HBH9 2/20 0.41
PRKCZ Q05513 2/20 0.38
ATR Q13535 1/20 0.36
PIM1 P11309 2/20 0.36
ROCK2 O75116 1/20 0.36
CDC42BPB Q9Y5S2 1/20 0.36
PIM3 Q86V86 1/20 0.35
PIM2 Q9P1W9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13442184 0.90 IKBKB (0.49) IKBKBCHUKROCK1LCKTNF
SCHEMBL13440925 0.89 IKBKB (0.53) IKBKBCHUKROCK1LCKTNF
SCHEMBL13442191 0.85 IKBKB (0.55) IKBKBCHUKROCK1LCKAKT1
SCHEMBL12326819 0.82 IKBKB (0.64) IKBKBCHUKROCK1LCKAKT1
SCHEMBL13087893 0.82 IKBKB (0.42) IKBKBCHUKROCK1LCKTNF
SCHEMBL13088170 0.82 IKBKB (0.44) IKBKBCHUKTNFATR
SCHEMBL13088196 0.82 IKBKB (0.53) IKBKBCHUKROCK1LCKTNF
SCHEMBL2424475 0.80 IKBKB (0.51) IKBKBCHUKROCK1LCKAKT1
SCHEMBL13440921 0.78 IKBKB (0.69) IKBKBCHUKROCK1LCKAKT1
SCHEMBL12327249 0.75 IKBKB (0.43) IKBKBCHUKROCK1LCKAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038465-A1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF 旭化成ファーマ株式会社 (JP) 2010-04-08 WO disclosed