SCHEMBL134424

SCHEMBL134424

CCOC(=O)Nc1cccc(OC(=O)Nc2cccc(C)c2)c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 5/20 0.77
ALDH1A1 P00352 2/20 0.77
CYP3A4 P08684 2/20 0.77
FAAH O00519 1/20 0.77
MTNR1B P49286 1/20 0.59
MAPT P10636 3/20 0.58
LMNA P02545 2/20 0.58
HSD17B10 Q99714 2/20 0.58
HTT P42858 2/20 0.54
NPC1 O15118 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
CYP1A2 P05177 3/20 0.53
CYP2C9 P11712 2/20 0.53
CYP2C19 P33261 2/20 0.53
GAA P10253 2/20 0.53
ALOX15 P16050 2/20 0.53
TSHR P16473 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HPGD P15428 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29512574 1.00 MAPK1 (0.77) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
Desmedipham SCHEMBL3230751 0.93 MAPK1 (0.79) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
Desmedipham SCHEMBL4659769 0.91 MAPK1 (0.75) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
Desmedipham SCHEMBL29516752 0.90 MAPK1 (0.68) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
Desmedipham SCHEMBL55084 0.90 MAPK1 (0.68) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
Desmedipham SCHEMBL4895813 0.90 MAPK1 (0.68) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
SCHEMBL3424143 0.90 MAPK1 (0.69) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
SCHEMBL11591205 0.90 ALDH1A1 (0.70) MAPK1ALDH1A1CYP3A4FAAHMTNR1B
Phenmedipham SCHEMBL54580 0.87 CYP3A4 (1.00) MAPK1ALDH1A1CYP3A4FAAHMAPT
Phenmedipham SCHEMBL8489570 0.87 CYP3A4 (1.00) MAPK1ALDH1A1CYP3A4FAAHMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5702 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260007133-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2026-01-08 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
US-20250268166-A1 ALS-INHIBITOR HERBICIDE TOLERANT BETA VULGARIS HYBRIDS WITH INCREASED HETEROSIS KWS SAAT SE & Co. KGaA (DE) 2025-08-28 US claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
US-12376586-B2 Microcapsules comprising cinmethyln in the core and a polyurea derived from diphenylmethane diisocyanate or an oligomer thereof BASF Agro B.V. (NL) 2025-08-05 US claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
EP-4554381-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2025-05-21 EP claimed
US-20240389528-A1 PERFORMANCE GAIN IN ALS INHIBITOR HERBICIDE TOLERANT BETA VULGARIS PLANTS BY COMBINATION OF BEST FITTING ALS LARGE AND SMALL SUBUNITS KWS SAAT SE & Co. KGaA (DE) 2024-11-28 US claimed
EP-3568016-B1 MICROCAPSULES COMPRISING CINMETHYLIN IN THE CORE AND A POLYUREA DERIVED FROM DIPHENYLMETHANE DIISOCYANATE OR AN OLIGOMER THEREOF BASF AGRO BV (NL) 2024-07-17 EP claimed
EP-1429609-B1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AG (DE) 2007-03-07 EP claimed
EP-1458237-B1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AG (DE) 2006-04-12 EP claimed
WO-2005058041-A2 METHOD FOR CONTROLLING CONIFEROUS PLANTS BASF AKTIENGESELLSCHAFT (DE) 2005-06-30 WO claimed
US-20050037923-A1 Herbicidal mixture based on 7-pyrazolybenzoxazoles BASF AKTIENGESELLSCHAFT (DE) 2005-02-17 US claimed
US-20040235665-A1 used in combination with other herbicides and possibly plant safening agents in order to reduce toxic effect on plants BASF AKTIENGESELLSCHAFT (DE) 2004-11-25 US claimed
EP-1458237-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2004-09-22 EP claimed
EP-1429609-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2004-06-23 EP claimed
WO-2003051122-A1 HERBICIDAL MIXTURE BASED ON 7-PYRAZOLYLBENZOXAZOLES BASF AKTIENGESELLSCHAFT (DE) 2003-06-26 WO claimed
WO-2003024221-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO claimed
EP-0102003-A1 Stabilised herbicide composition based on meta-biscarbamates S.I.P.C.A.M. S.p.A. Società Italiana Prodotti Chimici e per l'Agricoltura Milano (IT) 1984-03-07 EP claimed