Desmedipham

Desmedipham

SCHEMBL4895813

CCOC(=O)Nc1cccc(OC(=O)Nc2ccccc2)c1.CCOC(=O)Nc1cccc(OC(=O)Nc2ccccc2)c1

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.68
MAPT P10636 3/20 0.68
HSD17B10 Q99714 2/20 0.68
LMNA P02545 1/20 0.68
RAB9A P51151 3/20 0.65
HPGD P15428 2/20 0.65
NPC1 O15118 2/20 0.65
CRHBP P24387 1/20 0.65
CRHR2 Q13324 1/20 0.65
MTNR1B P49286 1/20 0.64
ALDH1A1 P00352 4/20 0.62
FAAH O00519 1/20 0.62
CYP3A4 P08684 1/20 0.62
KMT2A Q03164 1/20 0.61
BCHE P06276 1/20 0.60
ACHE P22303 1/20 0.60
CYP1A2 P05177 2/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
ALOX15 P16050 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Desmedipham SCHEMBL29516752 1.00 MAPK1 (0.68) MAPK1MAPTHSD17B10LMNARAB9A
Desmedipham SCHEMBL55084 1.00 MAPK1 (0.68) MAPK1MAPTHSD17B10LMNARAB9A
SCHEMBL4108576 0.93 MAPK1 (0.74) MAPK1MAPTHSD17B10LMNARAB9A
Desmedipham SCHEMBL725936 0.92 MAPT (0.59) MAPK1MAPTHSD17B10LMNARAB9A
Desmedipham SCHEMBL3230751 0.91 MAPK1 (0.79) MAPK1MAPTHSD17B10LMNARAB9A
SCHEMBL134424 0.90 MAPK1 (0.77) MAPK1MAPTHSD17B10LMNARAB9A
SCHEMBL29512574 0.90 MAPK1 (0.77) MAPK1MAPTHSD17B10LMNARAB9A
SCHEMBL11592554 0.89 ALDH1A1 (0.56) MAPK1MAPTHSD17B10LMNARAB9A
Desmedipham SCHEMBL4659769 0.89 MAPK1 (0.75) MAPK1MAPTHSD17B10LMNARAB9A
Desmedipham SCHEMBL28163042 0.89 FAAH (0.56) MAPK1MAPTHSD17B10LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 165 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3746505-B1 COMPOSITION, POLYMER COMPOSITE ARTICLE FORMED THEREWITH, AND METHOD OF PREPARING SAME DOW SILICONES CORP (US) 2024-06-26 EP disclosed
EP-3906245-B1 MULTIFUNCTIONAL ORGANOSILICON COMPOUND AND RELATED METHODS, COMPOUNDS, AND COMPOSITIONS DOW SILICONES CORP (US) 2024-05-29 EP disclosed
US-20240124709-A1 COMPOSITION, POLYMER COMPOSITE ARTICLE FORMED THEREWITH, AND METHOD OF PREPARING SAME DOW GLOBAL TECHNOLOGIES LLC 2024-04-18 US disclosed
EP-3645640-B1 SILICONE-POLYETHER COPOLYMER, METHOD OF PREPARING SAME, AND SEALANT COMPRISING SAME DOW SILICONES CORP (US) 2024-03-06 EP disclosed
US-11884821-B2 Composition, polymer composite article formed therewith, and method of preparing same DOW SILICONES CORPORATION (US) 2024-01-30 US disclosed
US-11807775-B2 Silicone-organic copolymer, sealants comprising same, and related methods DOW SILICONES CORPORATION (US) 2023-11-07 US disclosed
US-11760841-B2 Silicone-polycarbonate copolymer, sealants comprising same, and related methods DOW SILICONES CORPORATION (US) 2023-09-19 US disclosed
EP-3898779-B1 SILICONE-POLYESTER COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORP (US) 2023-02-08 EP disclosed
EP-3898781-B1 SILICONE-POLYCARBONATE COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORP (US) 2023-01-04 EP disclosed
US-20220064383-A1 SILICONE-POLYACRYLATE COPOLYMER, SEALANTS COMPRISING SAME, AND RELATED METHODS DOW SILICONES CORPORATION 2022-03-03 US disclosed
WO-2013013109-A1 GERMANIUM CONTAINING COMPLEX AND CONDENSATION REACTION CURABLE COMPOSITIONS AND METHODS FOR THE PREPARATION AND USE OF THE COMPOSITIONS DOW CORNING CORPORATION (US) 2013-01-24 WO disclosed
WO-2013009840-A1 LANTHANIDE COMPLEXES WITH IMIDAZOLE LIGANDS FOR CONDENSATION REACTIONS DOW CORNING CORPORATION (US) 2013-01-17 WO disclosed
WO-2013009836-A1 SAMARIUM CONTAINING COMPLEXES AND CONDENSATION REACTION CATALYSTS, METHODS FOR PREPARING THE CATALYSTS, AND COMPOSITIONS CONTAINING THE CATALYSTS DOW CORNING CORPORATION (US) 2013-01-17 WO disclosed
WO-2013000788-A1 HYDROSILYLATION REACTION CURABLE COMPOSITIONS AND METHODS FOR THEIR PREPARATION AND USE DOW CORNING CORPORATION (US) 2013-01-03 WO disclosed
WO-2012134784-A1 COMPOSITIONS CONTAINING PHOSPHONATE CATALYSTS AND METHODS FOR THE PREPARATION AND USE OF THE COMPOSITIONS DOW CORNING CORPORATION (US) 2012-10-04 WO disclosed
WO-2012134788-A1 COMPOSITIONS CONTAINING PHOSPHATE CATALYSTS AND METHODS FOR THE PREPARATION AND USE OF THE COMPOSITIONS DOW CORNING CORPORATION (US) 2012-10-04 WO disclosed
WO-2012134786-A1 COMPOSITIONS CONTINING SULFONIC ACID CATALYSTS AND METHODS FOR THE PREPARATION AND USE OF THE COMPOSITIONS DOW CORNING CORPORATION (US) 2012-10-04 WO disclosed
US-20080118734-A1 Coating Compositions DOW CORNING IRELAND LTD. (IE) 2008-05-22 US disclosed
EP-1744836-A2 PROCESS AND APPARATUS FOR PLASMA COATING, SUBSTRATES COATED BY THIS METHOD OR APPARATUS Dow Corning Ireland Limited (IE) 2007-01-24 EP disclosed
WO-2005110626-A2 PROCESS AND APPARATUS FOR PLASMA COATING, SUBSTRATES COATED BY THIS METOD OR APPARATUS DOW CORNING IRELAND LIMITED (IE) 2005-11-24 WO disclosed