SCHEMBL13445965

SCHEMBL13445965

Cc1ccc(S(=O)(=O)OCCOc2cccc(C(N)=O)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA9 Q16790 1/20 0.51
PARP1 P09874 2/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MAOB P27338 1/20 0.45
OPRM1 P35372 1/20 0.44
OPRD1 P41143 1/20 0.44
OPRK1 P41145 1/20 0.44
KCNH2 Q12809 1/20 0.44
POLB P06746 2/20 0.43
PARP10 Q53GL7 2/20 0.43
PRSS1 P07477 2/20 0.42
TNKS O95271 1/20 0.42
PARP15 Q460N3 1/20 0.42
PARP14 Q460N5 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL201311 0.93 PRSS1 (0.48) CA12CA1CA9PARP1KMT2A
SCHEMBL7390569 0.89 MAOB (0.59) CA12CA1CA9KMT2AMEN1
SCHEMBL21819012 0.89 KMT2A (0.57) CA12CA1CA9KMT2AMAOB
SCHEMBL31133435 0.89 KMT2A (0.57) CA12CA1CA9KMT2AMAOB
SCHEMBL29084505 0.87 TCF4 (0.53) CA12CA1CA9RAB9AMAOB
SCHEMBL29768638 0.87 TCF4 (0.53) CA12CA1CA9RAB9AMAOB
SCHEMBL29768570 0.84 TCF4 (0.50) CA12CA1CA9RAB9AMAOB
SCHEMBL13446449 0.82 CA12 (0.55) CA12CA1CA9KMT2AMEN1
SCHEMBL3071450 0.81 CA12 (0.56) CA12CA1CA9MAOBPOLB
SCHEMBL31408090 0.79 PAX8 (0.48) KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010028776-A1 PIPERAZINE DERIVATIVES FOR BINDING AND IMAGING AMYLOID PLAQUES AND THEIR USE BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-03-18 WO disclosed
EP-2163541-A1 Piperazine derivatives for binding and imaging amyloid plaques and their use Bayer Schering Pharma Aktiengesellschaft (DE) 2010-03-17 EP disclosed