SCHEMBL134467

SCHEMBL134467

CSc1c(N)nc(N)nc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 2/20 0.35
DPP4 P27487 1/20 0.34
HSP90AA1 P07900 3/20 0.34
MEN1 O00255 1/20 0.33
SLC22A1 O15245 1/20 0.33
ALDH1A1 P00352 1/20 0.33
DHFR P00374 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
HEXA P06865 1/20 0.33
HEXB P07686 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
HTR2A P28223 1/20 0.33
ADRA1A P35348 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30381851 1.00 HSP90AB1 (0.35) HSP90AB1DPP4HSP90AA1MEN1SLC22A1
SCHEMBL10990013 0.88 HSP90AB1 (0.39) HSP90AB1DPP4HSP90AA1HTR1AADORA2A
SCHEMBL10989493 0.82 CDK1 (0.32) ALDH1A1HTR1A
SCHEMBL10986250 0.77 HSP90AA1 (0.41) HSP90AA1MEN1SLC22A1ALDH1A1DHFR
SCHEMBL10984567 0.75 HTR1A (0.50) MEN1LMNACYP1A2HTR1AKMT2A
SCHEMBL10989049 0.75 PTPN1 (0.38) MEN1HTR1AKMT2A
SCHEMBL10982820 0.73 CDK1 (0.35) HSP90AB1ALDH1A1
SCHEMBL12463137 0.73 MAP4K4 (0.36) HSP90AB1HSP90AA1MEN1DHFRKMT2A
SCHEMBL10982815 0.72 APP (0.42) TDP1
SCHEMBL10987331 0.71 GAA (0.50) ALDH1A1LMNAHTR1AKMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3380 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
US-20210378241-A1 COMBINATION COMPRISING A BENZAMIDE HERBICIDE AND A PYRIDINE CARBOXYLIC ACID HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2021-12-09 US claimed
EP-3407717-B1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2021-07-28 EP claimed
CN-108697081-B Molecules having pesticidal utility, and intermediates, compositions and methods related thereto 美国陶氏益农公司 2021-07-23 CN claimed
EP-3407716-B9 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2021-07-14 EP claimed
EP-3407720-B1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2021-03-10 EP claimed
US-6632775-B1 Synergistic combination including a 3-aryl-1,3,4-thiadiazol-2(3H)-one; nonphytotoxic to agricultural crops ISAGRO RICERCA S.R.L. (IT) 2003-10-14 US claimed
EP-0986303-B1 HERBICIDAL COMPOSITIONS ISAGRO RICERCA SRL (IT) 2001-12-12 EP claimed
US-4528026-A 2-(Or4-)amino-5-alkylthio-pyrimidine herbicides PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1985-07-09 US claimed
EP-0080917-B1 HERBICIDAL COMPOSITIONS BASED ON 4-AMINO-6-CHLORO-5-ALKYLTHIO-PYRIMIDINE DERIVATIVES AND PYRIDATE, AND PROCESS FOR THE TREATMENT OF CORPS WITH THE AID OF SAID COMPOSITIONS P C U K PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1985-01-23 EP claimed
EP-0070219-B1 HERBICIDAL COMPOSITIONS BASED ON 4-AMINO-6-CHLORO-5-ALKYLTHIOPYRIMIDINE DERIVATIVES AND 2,6-DINITROANILINE DERIVATIVES, AND METHOD OF TREATING CROPS WITH SAID COMPOSITIONS P C U K PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1984-10-24 EP claimed
EP-0078623-A1 Herbicidal mixtures comprising benazolin FBC LIMITED (GB) 1983-05-11 EP claimed
EP-0033265-B1 HERBICIDAL COMPOSITIONS BASED ON 2,4-DIAMINO-6-CHLORO-5-METHYLTHIO-PYRIMIDINE AND DICLOFOP METHYL, AND PROCESS FOR THE TREATMENT OF CULTURES WITH THE AID OF SAID COMPOSITIONS P C U K PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1983-02-09 EP claimed
US-4359333-A AND 2,6-DIAMINO-2-CHLORO-5-METHYLTHIO PYRIMIDINE PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1982-11-16 US claimed
EP-0013636-B1 HERBICIDAL COMPOSITIONS CONTAINING 2,4-DIAMINO-6-CHLORO-5-METHYLTHIO-PYRIMIDINE AND HERBICIDAL UREA DERIVATIVES AND METHOD OF TREATMENT OF CULTURES WITH SAID COMPOSITIONS P C U K PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1982-02-24 EP claimed
EP-0000681-B1 AMINO-2 (OR -4) ALKYLTHIO-5 PYRIMIDINES, PROCESSES FOR THEIR PREPARATION, THEIR USE AS HERBICIDES AND COMPOSITION CONTAINING THEM P C U K PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1981-08-26 EP claimed