SCHEMBL134480

SCHEMBL134480

Nc1cnn(-c2ccccc2)c(=O)c1Br

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.70
SMN1; SMN2 Q16637 8/20 0.70
NPC1 O15118 7/20 0.70
ALDH1A1 P00352 6/20 0.70
LMNA P02545 4/20 0.70
MAPT P10636 4/20 0.70
HTT P42858 4/20 0.70
NPSR1 Q6W5P4 3/20 0.70
PAX8 Q06710 2/20 0.70
RXFP1 Q9HBX9 2/20 0.70
MAPK14 Q16539 1/20 0.55
KMT2A Q03164 4/20 0.54
POLB P06746 2/20 0.54
MEN1 O00255 3/20 0.52
XBP1 P17861 2/20 0.51
MITF O75030 1/20 0.51
S1PR4 O95977 1/20 0.51
THRB P10828 1/20 0.51
S1PR1 P21453 1/20 0.51
APP P05067 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10769084 0.83 RAB9A (0.71) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL11272238 0.83 RAB9A (0.51) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL27619397 0.83 RAB9A (0.70) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL4743412 0.82 RAB9A (1.00) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL10672542 0.82 RAB9A (0.58) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
Pyrazon SCHEMBL1858918 0.79 RAB9A (0.70) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
Pyrazon SCHEMBL53824 0.79 RAB9A (0.70) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL5842939 0.79 RAB9A (0.70) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL11285510 0.78 NPC1 (0.53) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA
SCHEMBL11098516 0.78 HIF1A (0.48) RAB9ASMN1; SMN2NPC1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3934 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
EP-3578541-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY, AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-05-28 EP claimed
US-20240130368-A1 HERBICIDAL COMPOSITION NIPPON SODA CO., LTD. (JP) 2024-04-25 US claimed
US-20240102976-A1 METHOD FOR SCREENING PESTICIDE RESIDUES IN MEDICINE FOOD HOMOLOGY CHARACTERISTIC AGRICULTUREAL PRODUCTS CHANGCHUN CUSTOMS TECHNOLOGY CENTER (CN) 2024-03-28 US claimed
EP-4316244-A1 HERBICIDAL COMPOSITION Nippon Soda Co., Ltd. (JP) 2024-02-07 EP claimed
CN-116867373-A Herbicidal composition 日本曹达株式会社 2023-10-10 CN claimed
US-20230139897-A1 SOLID HERBICIDE COMPOSITION AND THE USE THEREOF ROTAM AGROCHEM INTERNATIONAL COMPANY LIMITED (HK) 2023-05-04 US claimed
US-20230000079-A1 COMBINATION COMPRISING A TRIKETONE HERBICIDE AND A DIPHENYLETHER HERBICIDE, AND A METHOD FOR MAKING AND USING THE COMBINATION Generic Crop Science LLC (US) 2023-01-05 US claimed
EP-1313369-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2003-05-28 EP claimed
WO-2003024221-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO claimed
US-20020055435-A1 Herbicidal mixtures INTELLECTUAL PROPERTY DEPARTMENT (DE) 2002-05-09 US claimed
WO-2002015694-A2 HERBICIDAL MIXTURES BASF AKTIENGESELLSCHAFT (DE) 2002-02-28 WO claimed
US-4396415-A 1-PHENYL-4-AMINO-5-CHLORO (OR BROMO)PYRIDAZONE-6, PHENOLSULFONIC ACID-UREA-FORMALDEHYDE CONDENSATE, SILICA, ETHYLENE-OXIDE-PROPYLENE OXIDE COPOLYMER BASF AKTIENGESELLSCHAFT (DE) 1983-08-02 US claimed
EP-0017001-B1 HERBICIDES IN THE FORM OF AN AQUEOUS SUSPENSION CONTAINING A PYRIDAZONE AND A THIOLCARBAMATE, A CHLOROACETANILIDE OR A DINITROANILINE, AND A METHOD FOR THEIR PREPARATION AND ITS USE IN COMBATING UNDESIRED PLANT GROWTH BASF Aktiengesellschaft (DE) 1982-04-28 EP claimed
US-4305750-A Herbicides based on pyridazones BASF AKTIENGESELLSCHAFT (DE) 1981-12-15 US claimed
EP-0017001-A1 Herbicides in the form of an aqueous suspension containing a pyridazone and a thiolcarbamate, a chloroacetanilide or a dinitroaniline, and a method for their preparation and its use in combating undesired plant growth BASF Aktiengesellschaft (DE) 1980-10-15 EP claimed
US-4144048-A SYNERGISTIC MIXTURES BASF AKTIENGESELLSCHAFT (DE) 1979-03-13 US claimed
US-4021226-A 1-PHENYL-4-AMINO-5-CHLORO-PYRIDAZONE BASF AKTIENGESELLSCHAFT (DT) 1977-05-03 US claimed