SCHEMBL13448488

SCHEMBL13448488

C/C=C(C)\C(=N/C)c1cc(C)nc2c(OCc3c(Cl)cc(OC)nc3Cn3cccc(N)c3=O)cccc12

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 18/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C19 P33261 1/20 0.39
RORC P51449 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14038656 0.81 BDKRB2 (0.38) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12712319 0.81 BDKRB2 (0.42) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12711428 0.81 BDKRB2 (0.44) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12712424 0.80 BDKRB2 (0.39) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12712423 0.80 BDKRB2 (0.52) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13448486 0.79 BDKRB2 (0.48) BDKRB2CYP3A4CYP2C19
SCHEMBL13448512 0.79 BDKRB2 (0.52) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13448613 0.79 BDKRB2 (0.59) BDKRB2CYP3A4CYP2C19
SCHEMBL13093477 0.78 BDKRB2 (0.36) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13092954 0.77 BDKRB2 (0.39) BDKRB2CYP3A4CYP2C19RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010031589-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-03-25 WO disclosed