SCHEMBL13449018

SCHEMBL13449018

C[C@@H](c1ccc(C#N)cc1)n1cccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.45
CYP2A6 P11509 2/20 0.40
ALDH1A1 P00352 1/20 0.40
OPRD1 P41143 1/20 0.39
HSD11B1 P28845 2/20 0.39
CREBBP Q92793 1/20 0.39
TSHR P16473 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CYP2C19 P33261 1/20 0.38
CYP17A1 P05093 1/20 0.37
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DPP4 P27487 1/20 0.36
KCNH2 Q12809 1/20 0.36
GRIA1 P42261 1/20 0.36
GRIA2 P42262 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507790 0.78 CYP19A1 (0.71) CYP19A1CYP3A4CYP11B1CYP11B2CYP17A1
SCHEMBL12770872 0.74 CYP2D6 (0.54) ALDH1A1OPRD1CYP17A1KDM4EMAPT
SCHEMBL7009772 0.74 CYP2D6 (0.54) ALDH1A1OPRD1CYP17A1KDM4EMAPT
SCHEMBL12770874 0.74 CYP2D6 (0.54) ALDH1A1OPRD1CYP17A1KDM4EMAPT
SCHEMBL13962576 0.73 CYP2A6 (0.48) CYP19A1CYP2A6ALDH1A1TSHRCYP3A4
SCHEMBL7799578 0.72 CYP2A6 (0.52) CYP19A1CYP2A6ALDH1A1TSHRCYP3A4
SCHEMBL13557870 0.72 CYP2A6 (0.52) CYP19A1CYP2A6ALDH1A1TSHRCYP3A4
SCHEMBL87339 0.72 CYP2A6 (0.52) CYP19A1CYP2A6ALDH1A1TSHRCYP3A4
SCHEMBL6224919 0.72 SLC6A3 (0.50) CYP19A1CYP2A6ALDH1A1OPRD1HSD11B1
SCHEMBL20157572 0.70 TDP1 (0.45) HSD11B1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160196412-A1 DESIGN OF MOLECULES RECURSION PHARMACEUTICALS, INC. 2016-07-07 US disclosed
US-20120265514-A1 DESIGN OF MOLECULES UNIVERSITY OF DUNDEE (GB) 2012-10-18 US disclosed